Opiranserin hydrochloride

DESCRIPTION

Opiranserin (VVZ-149) hydrochloride is a dual antagonist of glycine transporter type 2 (GlyT2) and serotonin receptor 2A (5HT2A), with IC50s of 0.86 and 1.3 μM, respectively. It shows antagonistic activity on rP2X3 (IC50=0.87 μM). It is development as an injectable agent for the treatment of postoperative pain.

DETAILS

Cas: 1440796-75-7
Purity: 98.03%
Smiles: Cl.CCCCOc1c(OC)cc(cc1OC)C(=O)NCC1(CCOCC1)N(C)C
Category: Compound
Molecular Weight: 430.97
Molecular Formula: C21H35ClN2O5

Lead Time: < 1 week