(+)-MK-801 (hydrogen maleate)

DESCRIPTION

Potent, selective and non-competitive NMDA receptor antagonist (Ki = 30.5 nM); acts at the NMDA receptor-operated ion channel as an open channel blocker, preventing Ca2+ flux

DETAILS

Inchi: InChI=1S/C16H15N.C4H4O4/c1-16-13-8-4-2-6-11(13)10-15(17-16)12-7-3-5-9-14(12)16;5-3(6)1-2-4(7)8/h2-9,15,17H,10H2,1H3;1-2H,(H,5,6)(H,7,8)/b;2-1-/t15-,16+;/m1./s1
Purity: ≥98%
Raptas: Product Type|Biochemicals|Ion Channel Modulation|Blockers||Research Area|Neuroscience|Neuroprotection|Ischemia
Smiles: C[C@@]12C3=CC=CC=C3[C@@](N2)([H])CC4=CC=CC=C41.O=C(/C=C\C(O)=O)O
Inchikey: QLTXKCWMEZIHBJ-PJGJYSAQSA-N
Cas Number: 77086-22-7
Formulation: A crystalline solid
Item Origin: Synthetic
Storage Temp: -20
Shipping Temp: -20
Formula Markup: C16H15N • C4H4O4
Formula Weight: 337.4
Shelf Life Days: 1460