J-2156 TFA

DETAILS

Cas: 2387505-73-7
Purity: 98%
Smiles: OC(=O)C(F)(F)F.Cc1ccc(c2ccccc12)S(=O)(=O)N[C@@H](CCN)C(=O)N[C@@H](Cc1ccccc1)C(N)=O
Category: Compound
Molecular Weight: 582.6
Molecular Formula: C26H29F3N4O6S

DESCRIPTION

J-2156 TFA is a selective and potent growth inhibitor receptor type 4 (SST4) agonist that acts on the human SST4 receptor (IC50: 0.05 nM) and rat SST4 receptor (IC50: 0.07 nM). J-2156 TFA exhibited anti-inflammatory activity and was able to alleviate mechanical abnormal pain and mechanical hyperalgesia in the rat ipsilateral hind paw.

Lead Time: 4 - 5 weeks