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T38055

Salvinorin A Propionate

TargetMol

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DETAILS

  • Purity: 98%
  • Smiles: [H][C@@]12CC[C@@]3(C)[C@@H](C[C@H](OC(=O)CC)C(=O)[C@]3([H])[C@@]1(C)C[C@H](OC2=O)c1ccoc1)C(=O)OC
  • Category: Compounds
  • Cas Number: 689295-71-4
  • Molecular Weight: 446.496
  • Molecular Formula: C24H30O8

DESCRIPTION

Salvinorin A propionate is a selective partial agonist at κ1-opioid receptors (KOR) with a Ki value of 32.6 nM. It inhibits adenylate cyclase (EC50 = 4.7 nM) in HEK293 cells transfected with human KOR. It is selective for KORs over μ, δ, and ORL-1 opioid receptors and has no effect at serotonin, dopamine, muscarinic, or adrenergic receptors. In mice, salvinorin A propionate (13 μg, i.c.v.) reduces nociceptive responses in a radiant heat tail-flick assay, though not as potently as salvinorin A .

Lead Time: 4 - 5 weeks

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