PIK-75 hydrochloride

DETAILS

Cas: 372196-77-5
Purity: 98%
Smiles: Cc1ccc(cc1S(=O)(=O)N(C)/N=C/c1cnc2ccc(cn12)Br)[N+](=O)[O-].Cl
Category: Compound
Molecular Weight: 488.74
Molecular Formula: C16H14BrN5O4S·HCl

DESCRIPTION

PIK-75 hydrochloride (PIK-75 HCl) is a p110α inhibitor with IC50 of 5.8 nM (200-fold more potently than p110β), isoform-specific mutants at Ser773, and also potently inhibits DNA-PK with IC50 of 2 nM in cell-free assays.

Lead Time: 4 - 5 weeks