T28996
TP-064
TargetMol
DESCRIPTION
TP-064 is a potent and selective PRMT4 inhibitor. TP-064 includes inhibition of PRMT4 with IC50 < 10nM for methylation of H3 (1-25) and greater than 100-fold selectivity over other histone methyltransferases and non-epigenetic targets. TP-064 inhibits the methylation of MED12 with IC50 = 43 nM in cell.
DETAILS
- Cas: 2080306-20-1
- Purity: 99.07%
- Smiles: C(N(C(=O)C1=CC(OC2=CC=CC=C2)=CC=C1)C)C=3C=C(N=CC3)C4CCN(CCNC)CC4
- Category: Compound
- Molecular Weight: 458.6
- Molecular Formula: C28H34N4O2
Lead Time: 4 - 5 weeks
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