FTI-2153

DESCRIPTION:

FTI-2153 is a potent and highly selective farnesyltransferase (FTase) inhibitor (IC50: 1.4 nM) that is over 3000-fold more effective at blocking H-Ras (IC50: 10 nM) than Rap1A processing.

DETAILS

Cas: 344900-92-1
Purity: 98%
Smiles: COC(=O)[C@H](CCSC)NC(=O)c1ccc(CNCc2cnc[nH]2)cc1-c1ccccc1C
Category: Compound
Molecular Weight: 466.6
Molecular Formula: C25H30N4O3S

Lead Time: 5 + weeks